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Effect of Coadministered Rosuvastatin Systemic Exposure Coadministered drug and dosing Cyclosporine – stable dose required (75 mg – 200 mg BID) Gemfibrozil 600 mg BID for 7 days Lopinavir/ritonavir combination 400 mg/100 mg BID for 10 days Atazanavir/ritonavir combination 300 mg/100 mg QD for 7 days Tipranavir/ritonavir combination 500 mg/200mg BID for 11 days Fosamprenavir/ritonavir 700 mg/100 mg BID for 7 days Fenofibrate 67 mg TID for 7 days Aluminum & magnesium hydroxide combination antacid Administered simultaneously Administered 2 hours apart Erythromycin 500 mg QID for 7 days Ketoconazole 200 mg BID for 7 days Itraconazole 200 mg QD for 5 days Fluconazole 200 mg QD for 11 days *Single dose unless otherwise noted Mean crestor 50mg is rosuvastatin calcium as good as crestor crestor side effects alcohol rosuvastatin or ratio (with/without coadministered drug and no change = 1-fold) or % change (with/without coadministered drug and no change = 0%); symbols of ↑ and ↓ indicate the exposure increase and decrease, respectively .
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